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Open Access
Peer-reviewed
Research Article
A Potent Class of GPR40 Full Agonists Engages the EnteroInsular Axis to Promote Glucose Control in Rodents
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Jian Luo ,
Contributed equally to this work with: Jian Luo, Gayathri Swaminath
Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America
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Gayathri Swaminath ,
Contributed equally to this work with: Jian Luo, Gayathri Swaminath
Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America
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Sean P. Brown,
Affiliation Department of Therapeutic Discovery, Amgen Inc., South San Francisco, California, United States of America
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Jane Zhang,
Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America
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Qi Guo,
Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America
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Michael Chen,
Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America
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Kathy Nguyen,
Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America
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Thanhvien Tran,
Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America
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Lynn Miao,
Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America
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Paul J. Dransfield,
Affiliation Department of Therapeutic Discovery, Amgen Inc., South San Francisco, California, United States of America
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Marc Vimolratana,
Affiliation Department of Therapeutic Discovery, Amgen Inc., South San Francisco, California, United States of America
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Jonathan B. Houze,
Affiliation Department of Therapeutic Discovery, Amgen Inc., South San Francisco, California, United States of America
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Simon Wong,
Affiliation Department of Pharmacokinetics and Drug Metabolism, Amgen Inc., South San Francisco, California, United States of America
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Maria Toteva,
Affiliation Department of Pharmaceutics, Amgen Inc., South San Francisco, California, United States of America
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Bei Shan,
Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America
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Frank Li,
Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America
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Run Zhuang,
Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America
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Daniel C.-H. Lin
* E-mail: dclin@amgen.com
Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America
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A Potent Class of GPR40 Full Agonists Engages the EnteroInsular Axis to Promote Glucose Control in Rodents
- Jian Luo,
- Gayathri Swaminath,
- Sean P. Brown,
- Jane Zhang,
- Qi Guo,
- Michael Chen,
- Kathy Nguyen,
- Thanhvien Tran,
- Lynn Miao,
- Paul J. Dransfield
- Published: October 9, 2012
- https://doi.org/10.1371/journal.pone.0046300