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Discovery of Diverse Small Molecule Chemotypes with Cell-Based PKD1 Inhibitory Activity

  • Elizabeth R. Sharlow ,

    ers7g@virginia.edu

    Affiliation Department of Pharmacology, University of Virginia, Charlottesville, Virginia, United States of America

  • Gabriela Mustata Wilson,

    Affiliations Department of Computational and Systems Biology, University of Pittsburgh, Pittsburgh, Pennsylvania, United States of America, Drug Discovery Institute, University of Pittsburgh, Pittsburgh, Pennsylvania, United States of America

  • David Close,

    Affiliations Drug Discovery Institute, University of Pittsburgh, Pittsburgh, Pennsylvania, United States of America, Department of Pharmacology and Chemical Biology, University of Pittsburgh, Pittsburgh, Pennsylvania, United States of America

  • Stephanie Leimgruber,

    Affiliations Drug Discovery Institute, University of Pittsburgh, Pittsburgh, Pennsylvania, United States of America, Department of Pharmacology and Chemical Biology, University of Pittsburgh, Pittsburgh, Pennsylvania, United States of America

  • Manuj Tandon,

    Affiliation Department of Pharmacology and Chemical Biology, University of Pittsburgh, Pittsburgh, Pennsylvania, United States of America

  • Robyn B. Reed,

    Affiliations Drug Discovery Institute, University of Pittsburgh, Pittsburgh, Pennsylvania, United States of America, Department of Pharmacology and Chemical Biology, University of Pittsburgh, Pittsburgh, Pennsylvania, United States of America

  • Tong Ying Shun,

    Affiliations Drug Discovery Institute, University of Pittsburgh, Pittsburgh, Pennsylvania, United States of America, Department of Pharmacology and Chemical Biology, University of Pittsburgh, Pittsburgh, Pennsylvania, United States of America

  • Q. Jane Wang,

    Affiliations Drug Discovery Institute, University of Pittsburgh, Pittsburgh, Pennsylvania, United States of America, Department of Pharmacology and Chemical Biology, University of Pittsburgh, Pittsburgh, Pennsylvania, United States of America

  • Peter Wipf,

    Affiliations Drug Discovery Institute, University of Pittsburgh, Pittsburgh, Pennsylvania, United States of America, Department of Chemistry, University of Pittsburgh, Pittsburgh, Pennsylvania, United States of America

  • John S. Lazo

    Affiliations Department of Pharmacology, University of Virginia, Charlottesville, Virginia, United States of America, Department of Chemistry, University of Virginia, Charlottesville, Virginia, United States of America

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