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Modifying Ligand-Induced and Constitutive Signaling of the Human 5-HT4 Receptor

  • Wei Chun Chang,

    Current address: Lexicon Pharmaceuticals, The Woodlands, Texas, United States of America

    Affiliations Gladstone Institute of Cardiovascular Disease, University of California at San Francisco, San Francisco, California, United States of America, Graduate Program in Pharmaceutical Sciences and Pharmacogenomics, University of California at San Francisco, San Francisco, California, United States of America

  • Jennifer K. Ng,

    Affiliation Gladstone Institute of Cardiovascular Disease, University of California at San Francisco, San Francisco, California, United States of America

  • Trieu Nguyen,

    Affiliation Gladstone Institute of Cardiovascular Disease, University of California at San Francisco, San Francisco, California, United States of America

  • Lucie Pellissier,

    Affiliations Institut de Génomique Fonctionnelle, Universités de Montpellier, CNRS UMR 5203, Montpellier, France, INSERM U661, Montpellier, France

  • Sylvie Claeysen,

    Affiliations Institut de Génomique Fonctionnelle, Universités de Montpellier, CNRS UMR 5203, Montpellier, France, INSERM U661, Montpellier, France

  • Edward C. Hsiao,

    Affiliations Gladstone Institute of Cardiovascular Disease, University of California at San Francisco, San Francisco, California, United States of America, Department of Medicine, University of California at San Francisco, San Francisco, California, United States of America

  • Bruce R. Conklin

    To whom correspondence should be addressed. E-mail: bconklin@gladstone.ucsf.edu

    Affiliations Gladstone Institute of Cardiovascular Disease, University of California at San Francisco, San Francisco, California, United States of America, Department of Medicine, University of California at San Francisco, San Francisco, California, United States of America, Department of Cellular and Molecular Pharmacology, University of California at San Francisco, San Francisco, California, United States of America

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