About the Authors

John C. Castle

Contributed equally to this work with: John C. Castle, Yoshikazu Hara

john_castle@merck.com (JCC); jason_johnson@merck.com (JMJ)

Affiliation Rosetta Inpharmatics LLC, Seattle, Washington, United States of America

Yoshikazu Hara

Contributed equally to this work with: John C. Castle, Yoshikazu Hara

Affiliation Metabolic Disorder Research, Tsukuba Research Institute, Banyu Pharmaceutical Co., Ltd., Tsukuba, Ibaraki, Japan

Christopher K. Raymond

Affiliation Rosetta Inpharmatics LLC, Seattle, Washington, United States of America

Philip Garrett-Engele

Affiliation Rosetta Inpharmatics LLC, Seattle, Washington, United States of America

Kenji Ohwaki

Affiliation Metabolic Disorder Research, Tsukuba Research Institute, Banyu Pharmaceutical Co., Ltd., Tsukuba, Ibaraki, Japan

Zhengyan Kan

Affiliation Rosetta Inpharmatics LLC, Seattle, Washington, United States of America

Jun Kusunoki

Affiliation Metabolic Disorder Research, Tsukuba Research Institute, Banyu Pharmaceutical Co., Ltd., Tsukuba, Ibaraki, Japan

Jason M. Johnson

john_castle@merck.com (JCC); jason_johnson@merck.com (JMJ)

Affiliation Rosetta Inpharmatics LLC, Seattle, Washington, United States of America

Competing Interests

The authors have declared that no competing interests exist.

Author Contributions

Conceived and designed the experiments: JC CR KO JK JMJ. Performed the experiments: YH CR PGE KO. Analyzed the data: JC YH CR KO ZK. Contributed reagents/materials/analysis tools: JC CR PGE KO. Wrote the paper: JC CR KO JK JMJ.