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A Potent Class of GPR40 Full Agonists Engages the EnteroInsular Axis to Promote Glucose Control in Rodents

  • Jian Luo ,

    Contributed equally to this work with: Jian Luo, Gayathri Swaminath

    Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America

  • Gayathri Swaminath ,

    Contributed equally to this work with: Jian Luo, Gayathri Swaminath

    Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America

  • Sean P. Brown,

    Affiliation Department of Therapeutic Discovery, Amgen Inc., South San Francisco, California, United States of America

  • Jane Zhang,

    Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America

  • Qi Guo,

    Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America

  • Michael Chen,

    Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America

  • Kathy Nguyen,

    Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America

  • Thanhvien Tran,

    Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America

  • Lynn Miao,

    Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America

  • Paul J. Dransfield,

    Affiliation Department of Therapeutic Discovery, Amgen Inc., South San Francisco, California, United States of America

  • Marc Vimolratana,

    Affiliation Department of Therapeutic Discovery, Amgen Inc., South San Francisco, California, United States of America

  • Jonathan B. Houze,

    Affiliation Department of Therapeutic Discovery, Amgen Inc., South San Francisco, California, United States of America

  • Simon Wong,

    Affiliation Department of Pharmacokinetics and Drug Metabolism, Amgen Inc., South San Francisco, California, United States of America

  • Maria Toteva,

    Affiliation Department of Pharmaceutics, Amgen Inc., South San Francisco, California, United States of America

  • Bei Shan,

    Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America

  • Frank Li,

    Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America

  • Run Zhuang,

    Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America

  •  [ ... ],
  • Daniel C.-H. Lin

    dclin@amgen.com

    Affiliation Department of Metabolic Disorders, Amgen Inc., South San Francisco, California, United States of America

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