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Design, Synthesis and Characterization of a Highly Effective Inhibitor for Analog-Sensitive (as) Kinases

  • Michael Klein,

    Affiliation Medicinal Chemistry, Department of Chemistry, University of Gothenburg, Göteborg, Sweden

  • Montse Morillas,

    Affiliation Cell Signalling Unit, Department de Ciències Experimentals i de la Salut, Universitat Pompeu Fabra (UPF), Parc de Recerca Biomèdica de Barcelona (PRBB), Barcelona, Spain

  • Alexandre Vendrell,

    Affiliation Cell Signalling Unit, Department de Ciències Experimentals i de la Salut, Universitat Pompeu Fabra (UPF), Parc de Recerca Biomèdica de Barcelona (PRBB), Barcelona, Spain

  • Lars Brive,

    Affiliation Department of Cell and Molecular Biology, University of Gothenburg, Göteborg, Sweden

  • Marinella Gebbia,

    Affiliation Department of Pharmaceutical Sciences, University of Toronto, Toronto, Canada

  • Iain M. Wallace,

    Affiliation Department of Pharmaceutical Sciences, University of Toronto, Toronto, Canada

  • Guri Giaever,

    Affiliation Department of Pharmaceutical Sciences, University of Toronto, Toronto, Canada

  • Corey Nislow,

    Affiliation Department of Molecular Genetics, University of Toronto, Toronto, Canada

  • Francesc Posas,

    Affiliation Cell Signalling Unit, Department de Ciències Experimentals i de la Salut, Universitat Pompeu Fabra (UPF), Parc de Recerca Biomèdica de Barcelona (PRBB), Barcelona, Spain

  • Morten Grøtli

    grotli@chem.gu.se

    Affiliation Medicinal Chemistry, Department of Chemistry, University of Gothenburg, Göteborg, Sweden

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